KEGG DGROUP: CYP2D6 substrate
Lafutidine (JP18/INN) <JP>
Vonoprazan
Vonoprazan (USAN/INN)
Vonoprazan fumarate (JAN/USAN) <JP/US>
Vonoprazan, amoxicillin and clarithromycin <JP>
Vonoprazan, amoxicillin and metronidazole <JP>
Metoclopramide
Metoclopramide (JP18/INN) <JP>
Metoclopramide hydrochloride (JAN) <JP>
Metoclopramide hydrochloride (USP) <US>
Ondansetron
Ondansetron (JAN/USP/INN) <US>
Ondansetron hydrochloride hydrate (JAN/USP) <JP/US>
Dolasetron
Dolasetron (INN)
Dolasetron mesylate (USP)
Palonosetron
Palonosetron (INN)
Palonosetron hydrochloride (JAN/USP) <JP/US>
Fosnetupitant and palonosetron hydrochloride <US>
Fenfluramine
Fenfluramine (INN)
Fenfluramine hydrochloride (JAN/USAN) <JP/US>
Dexfenfluramine
Dexfenfluramine (INN)
Dexfenfluramine hydrochloride (USAN)
Phenformin
Phenformin (BAN)
Phenformin hydrochloride
Eliglustat
Eliglustat (USAN/INN)
Eliglustat tartrate (JAN/USAN) <JP/US>
Cilostazol (JP18/USP/INN) <JP/US>
Sparteine
Sparteine (INN)
Sparteine sulfate (JAN/USAN)
Ajmaline (JP18)
Mexiletine
Mexiletine (INN)
Mexiletine hydrochloride (JP18/USP) <JP/US>
Aprindine
Aprindine (USAN/INN)
Aprindine hydrochloride (JP18/USAN) <JP>
Propafenone
Propafenone (INN)
Propafenone hydrochloride (JP18/USP) <JP/US>
Flecainide
Flecainide (INN)
Flecainide acetate (JP18/USP) <JP/US>
Encainide
Encainide (INN)
Encainide hydrochloride (USAN)
Cibenzoline
Cifenline (USAN); Cibenzoline (INN)
Cifenline succinate (USAN); Cibenzoline succinate (JP18) <JP>
Urapidil
Urapidil (JP18/INN) <JP>
Urapidil hydrochloride
Debrisoquin sulfate (USAN)
Alprenolol
Alprenolol (INN)
Alprenolol hydrochloride (JP18/USAN)
Pindolol (JP18/USP/INN) <JP/US>
Propranolol
Propranolol (INN)
Propranolol hydrochloride (JP18/USP) <JP/US>
Timolol
Timolol (INN)
Timolol (USAN) <US>
Timolol maleate (JP18/USP) <JP/US>
Carteolol
Carteolol (INN)
Carteolol hydrochloride (JP18/USP) <JP/US>
Bopindolol
Bopindolol (INN)
Bopindolol malonate (JAN)
Metoprolol
Metoprolol (USAN/INN)
Metoprolol tartrate (JP18/USP) <JP/US>
Metoprolol succinate (USP) <US>
Metoprolol fumarate (USP)
Atenolol (JP18/USP/INN) <JP/US>
Nebivolol
Nebivolol (USAN/INN)
Nebivolol hydrochloride (USAN) <US>
Carvedilol
Carvedilol (JP18/USP/INN) <JP/US>
Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN) <US>
Metoprolol and hydrochlorothiazide <US>
Bepridil
Bepridil (INN)
Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN) <JP>
Perhexiline
Perhexiline (INN)
Perhexiline maleate (USAN)
Promethazine
Promethazine (JAN/INN)
Promethazine hydrochloride (JP18/USP) <JP/US>
Promethazine teoclate (JAN/INN)
Promethazine methylenedisalicylate (JAN) <JP>
Promethazine maleate
Promethazine hibenzate <JP>
Doxepin
Doxepin (INN)
Doxepin hydrochloride (USP) <US>
Tolterodine
Tolterodine (USAN/INN)
Tolterodine tartrate (JAN/USP) <JP/US>
Darifenacin
Darifenacin (USAN/INN)
Darifenacin hydrobromide (JAN/USAN) <US>
Fesoterodine
Fesoterodine (INN)
Fesoterodine fumarate (JAN/USAN) <JP/US>
Dutasteride and tamsulosin <US>
Elagolix, estradiol and norethisterone <US>
Osilodrostat
Osilodrostat (USAN/INN)
Osilodrostat phosphate (JAN/USAN) <JP/US>
Telithromycin (JAN/USAN/INN)
Delamanid (JAN/USAN) <JP>
Ritonavir (JAN/USP/INN) <JP/US>
Nevirapine (JAN/USP/INN) <JP/US>
Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil
Darunavir and cobicistat <JP/US>
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide <JP/US>
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide <JP/US>
Vorasidenib
Vorasidenib (USAN/INN)
Vorasidenib citrate (USAN); Vorasidenib citric acid hydrate (JAN) <US>
Nirogacestat
Nirogacestat (USAN/INN)
Nirogacestat hydrobromide (USAN) <US>
Tamoxifen
Tamoxifen (INN)
Tamoxifen citrate (JP18/USP) <JP/US>
Mavorixafor (USAN) <US>
Upadacitinib
Upadacitinib (USAN/INN)
Upadacitinib tartrate (USAN)
Upadacitinib hydrate (JAN) <JP/US>
Deucravacitinib (JAN/USAN) <JP/US>
Iptacopan
Iptacopan (USAN/INN)
Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN) <JP/US>
Pirfenidone (JAN/USAN/INN) <JP/US>
Oxycodone
Oxycodone (USAN/INN) <US>
Oxycodone hydrochloride (USP) <US>
Compound oxycodone (JP18)
Oxycodone terephthalate (USP)
Oxycodone hydrochloride hydrate (JP18) <JP>
Dihydrocodeine
Dihydrocodeine (INN)
Dihydrocodeine phosphate (JP18) <JP>
Dihydrocodeine bitartrate (USP)
Dihydrocodeine thiocyanate
dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea <JP>
Tramadol hydrochloride and acetaminophen <JP/US>
Tramadol
Tramadol (INN)
Tramadol hydrochloride (JP18/USP) <JP/US>
Naratriptan
Naratriptan (INN)
Naratriptan hydrochloride (JAN/USP) <JP/US>
Almotriptan
Almotriptan (USAN)
Almotriptan malate (USP) <US>
Ganaxolone (USAN/INN) <US>
Selegiline
Selegiline (USAN/INN) <US>
Selegiline hydrochloride (JAN/USP) <JP/US>
Chlorpromazine
Chlorpromazine (USP/INN)
Chlorpromazine hydrochloride (JP18/USP) <JP/US>
Chlorpromazine hibenzate (JAN)
Chlorpromazine phenolphthalinate (JAN) <JP>
Chlorpromazine tannate (JAN)
Fluphenazine
Fluphenazine (INN)
Fluphenazine hydrochloride (JAN/USP) <US>
Fluphenazine enanthate (JP18/USP)
Fluphenazine decanoate (JAN/USP) <JP/US>
Fluphenazine maleate (JAN) <JP>
Perphenazine
Perphenazine (JP18/USP/INN) <JP/US>
Perphenazine maleate (JP18) <JP>
Perphenazine fendizoate (JAN) <JP>
Perphenazine hydrochloride <JP>
Perphenazine decanoate
Perphenazine enantate
Haloperidol
Haloperidol (JP18/USP/INN) <JP/US>
Haloperidol decanoate (JAN/USP) <JP/US>
Haloperidol lactate <US>
Zuclopenthixol
Zuclopenthixol (INN)
Zuclopenthixol acetate
Zuclopenthixol decanoate
Zuclopenthixol dihydrochloride
Pimozide (JP18/USP/INN) <US>
Loxapine
Loxapine (USAN/INN) <US>
Loxapine succinate (USP) <US>
Loxapine hydrochloride
Olanzapine
Olanzapine (JAN/USP/INN) <JP/US>
Olanzapine pamoate (USAN) <US>
Risperidone (JP18/USP/INN) <JP/US>
Aripiprazole
Aripiprazole (JP18/USP/INN) <JP/US>
Aripiprazole cavoxil (USAN)
Aripiprazole lauroxil (USAN) <US>
Aripiprazole hydrate (JAN) <JP/US>
Iloperidone (USAN/INN) <US>
Cariprazine
Cariprazine (USAN/INN)
Cariprazine hydrochloride (JAN/USAN) <US>
Brexpiprazole (JAN/USAN/INN) <JP/US>
Pimavanserin tartrate (USAN) <US>
Chlorpromazine hydrochloride, promethazine hydrochloride and phenobarbital
Dexmedetomidine
Dexmedetomidine (USAN/INN)
Dexmedetomidine hydrochloride (JAN/USP) <JP/US>
Imipramine
Imipramine (INN)
Imipramine hydrochloride (JP18/USP) <JP/US>
Imipramine pamoate (USP) <US>
Clomipramine
Clomipramine (INN)
Clomipramine hydrochloride (JP18/USP) <JP/US>
Amitriptyline
Amitriptyline (INN)
Amitriptyline hydrochloride (JP18/USP) <JP/US>
Nortriptyline
Nortriptyline (INN)
Nortriptyline hydrochloride (JP18/USP/INN) <JP/US>
Dosulepin
Dosulepin (INN)
Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN) <JP>
Amoxapine (JP18/USP/INN) <JP/US>
Maprotiline
Maprotiline (USAN)
Maprotiline hydrochloride (JP18/USP) <JP>
Fluoxetine
Fluoxetine (USAN/INN)
Fluoxetine hydrochloride (JAN/USP) <US>
Citalopram
Citalopram (USP/INN)
Citalopram hydrobromide (USP) <US>
Citalopram hydrochloride
Paroxetine
Paroxetine (USP/INN)
Paroxetine hydrochloride hemihydrate (USP); Paroxetine hydrochloride hydrate (JP18) <JP/US>
Paroxetine hydrochloride (USP) <US>
Paroxetine mesylate (USAN) <US>
Fluvoxamine
Fluvoxamine (INN)
Fluvoxamine maleate (JP18/USP) <JP/US>
Escitalopram
Escitalopram (INN)
Escitalopram oxalate (JAN/USP) <JP/US>
Mianserin
Mianserin (INN)
Mianserin hydrochloride (JAN/USAN) <JP>
Trazodone
Trazodone (INN)
Trazodone hydrochloride (JAN/USP) <JP/US>
Minaprine
Minaprine (USAN/INN)
Minaprine hydrochloride (USAN)
Viloxazine
Viloxazine (INN)
Viloxazine hydrochloride (USAN) <US>
Mirtazapine
Mirtazapine (JAN/USP/INN) <JP/US>
Mirtazapine hydrate (JAN)
Venlafaxine
Venlafaxine (INN)
Venlafaxine hydrochloride (JAN/USP) <JP/US>
Venlafaxine besylate monohydrate <US>
Duloxetine
Duloxetine (INN)
Duloxetine hydrochloride (JAN/USP) <JP/US>
Vilazodone
Vilazodone (USAN/INN)
Vilazodone hydrochloride (USAN) <US>
Vortioxetine
Vortioxetine (USAN)
Vortioxetine hydrobromide (JAN/USAN) <JP/US>
Vortioxetine hemihydrobromide (USAN)
Dextromethorphan hydrobromide and bupropion hydrochloride <US>
Cinnarizine
Cinnarizine (JAN/USAN/INN)
Cinnarizine dihydrochloride
Amfetamine
Amfetamine (INN) <US>
Amphetamine sulfate (USP) <US>
Dexamfetamine
Dextroamphetamine (USAN); Dexamfetamine (INN) <US>
Dextroamphetamine sulfate (USP) <US>
Methamphetamine
Metamfetamine (INN)
Methamphetamine hydrochloride (JP18/USP) <JP/US>
Atomoxetine
Atomoxetine (USP/INN)
Atomoxetine hydrochloride (JAN/USP) <JP/US>
Donepezil
Donepezil (JAN/INN) <JP>
Donepezil hydrochloride (JP18/USP) <JP/US>
Galantamine
Galantamine (USAN/INN)
Galantamine hydrobromide (JAN/USP) <JP/US>
Cevimeline
Cevimeline (INN)
Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN) <JP/US>
Methadone
Methadone (BAN)
Methadone hydrochloride (JAN/USP) <JP/US>
Flunarizine
Flunarizine (INN)
Flunarizine hydrochloride (JAN/USAN)
Tetrabenazine (JAN/INN) <JP/US>
Pitolisant
Pitolisant (USAN/INN)
Pitolisant hydrochloride (USAN) <US>
Valbenazine
Valbenazine (USAN/INN)
Valbenazine tosylate (USAN); Valbenazine tosilate (JAN) <JP/US>
Umeclidinium bromide and vilanterol <JP/US>
Hydrocodone
Hydrocodone (INN)
Hydrocodone bitartrate (USP) <US>
Hydrocodone polistirex (USAN)
Hydrocodone hydrochloride
Codeine
Codeine
Codeine (USP)
Codeine phosphate (USP); Codeine phosphate hydrate (JP18) <JP>
Codeine polistirex (USAN)
Codeine sulfate (USP) <US>
Codeine hydrochloride
Dextromethorphan
Dextromethorphan (USP)
Dextromethorphan hydrobromide (USP); Dextromethorphan hydrobromide hydrate (JP18) <JP>
Dextromethorphan polistirex (USAN)
Codeine phosphate and chlorpheniramine maleate <US>
Dextromethorphan hydrobromide and potassium cresolsulfonate <JP>
Dexchlorpheniramine
Dexchlorpheniramine (INN)
Dexchlorpheniramine maleate (USP); d-Chlorpheniramine maleate (JP18) <JP/US>
Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate <JP>
Chlorpheniramine polistirex and codeine polistirex
Mequitazine (JP18/INN) <JP>
Loratadine (JAN/USP/INN) <JP/US>
Brinzolamide and timolol maleate <JP>
Dorzolamide hydrochloride and timolol maleate (JP18) <JP/US>
Cobicistat (JAN/USAN/INN) <US>
Ramosetron
Ramosetron (INN)
Ramosetron hydrochloride (JAN) <JP>
Umeclidinium
Umeclidinium (USAN)
Umeclidinium bromide (JAN/USAN) <JP/US>
Trelagliptin
Trelagliptin (USAN)
Trelagliptin succinate (JAN/USAN) <JP>
Sarpogrelate
Sarpogrelate (INN)
Sarpogrelate hydrochloride (JP18) <JP>
Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride <JP>
Sofpironium bromide (JAN/USAN/INN) <JP/US>
Butalbital, acetaminophen, caffeine and codeine phosphate <US>
Butalbital, aspirin, caffeine and codeine <US>
Vonoprazan and amoxicillin <US>
Xanomeline and trospium chloride <US>
Benzhydrocodone
Benzhydrocodone (USAN/INN)
Benzhydrocodone hydrochloride (USAN)
Bunitrolol hydrochloride (JAN)
Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate
Benzhydrocodone and acetaminophen <US>